DOAJ Open Access 2021

A noncanonical AR addiction drives enzalutamide resistance in prostate cancer

Yundong He Ting Wei Zhenqing Ye Jacob J. Orme Dong Lin +10 lainnya

Abstrak

Resistance to second generation anti-androgen therapies such as enzalutamide (ENZ) can emerge in prostate cancer patients. Here, the authors identify an ENZ-resistant mechanism driven by AR-dependent transcription of noncanonical targets that make resistant cells susceptible to dual inhibition of BET and CBP/p300 signaling.

Topik & Kata Kunci

Penulis (15)

Y

Yundong He

T

Ting Wei

Z

Zhenqing Ye

J

Jacob J. Orme

D

Dong Lin

H

Haoyue Sheng

L

Ladan Fazli

R

R. Jeffrey Karnes

R

Rafael Jimenez

L

Liguo Wang

L

Liewei Wang

M

Martin E. Gleave

Y

Yuzhuo Wang

L

Lei Shi

H

Haojie Huang

Format Sitasi

He, Y., Wei, T., Ye, Z., Orme, J.J., Lin, D., Sheng, H. et al. (2021). A noncanonical AR addiction drives enzalutamide resistance in prostate cancer. https://doi.org/10.1038/s41467-021-21860-7

Akses Cepat

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Informasi Jurnal
Tahun Terbit
2021
Sumber Database
DOAJ
DOI
10.1038/s41467-021-21860-7
Akses
Open Access ✓